產(chǎn)品編號 | D58240 |
英文名稱 | Calmidazolium chloride |
中文名稱 | 鈣調(diào)蛋白抑制劑 |
別 名 | R 24571 |
CAS | 57265-65-3 |
理論分子量 | 687.7kDa |
保存條件 | Powder: -20℃ for 3 years | In solvent: -80℃ for 1 year |
產(chǎn)品介紹 |
Calmidazolium chloride is a calmodulin (CaMK) antagonist (Kd = 3 nM), antagonizing CaM-dependent phosphodiesterase(IC50 = 0.15 μM) and calmodulin-induced activation of erythrocyte Ca2+-transporting ATPase(IC50 = 0.35 μM). Calmidazolium chloride also induces apoptosis in certain cancer cell lines. |